progestogenic การใช้

• Note that testosterone itself does not have significant progestogenic activity.
• Its analogue, SC-5233, possesses similar but less potent progestogenic activity.
• In addition to its progestogenic activity, NET also has weak androgenic and estrogenic effects at high dosages.
• In addition, along with SC-8109, it has been found to possess potent progestogenic activity.
• Cyproterone has approximately one-third the potency of CPA as an antiandrogen and is devoid of progestogenic activity.
• MPA has also been prescribed in male-to-female transgender individuals due to its progestogenic and antigonadotropic effects.
• Also unlike CPA, due to its lack of progestogenic and antigonadotropic activity, cyproterone does not suppress ovulation in women.
• Bolandiol ( and its dipropionate ester ) is unique among AAS in that it reportedly also possesses estrogenic and progestogenic activity.
• Note that while nandrolone ( 19-nortestosterone ) does have significant progestogenic activity, it is not used as a progestogen.
• Experience from experimental aromatase inhibitor treatment of endometriosis indicates that aromatase inhibitors might be particularly useful in combination with a progestogenic ovulation inhibitor.
• Similarly to nandrolone, dimethandrolone, and other 19-nortestosterone derivatives, 11?-MNT has been found to possess progestogenic activity.
• In addition to its antimineralocorticoid activity, SC-8109 shows potent progestogenic activity, with similar potency relative to that of progesterone.
• In addition to its glucocorticoid activity, mometasone also has very potent progestogenic activity and acts as a partial agonist of the mineralocorticoid receptor.
• "' Medrysone "'( structure to progesterone, neither progestogenic nor androgenic activity has been demonstrated for or attributed to medrysone.
• In contrast, 9?-fluoro-11?-hydroxyprogesterone has much lower progestogenic activity with only about 8 times that of 11?-hydroxyprogesterone.
• It was indicated as an oral treatment for prevention of estrus ( heat ) in adult female dogs . although potent and significant progestogenic activity remains present.
• Due to its progestogenic ( and by extension antigonadotropic ) activity, is able to suppress circulating testosterone levels by 70 80 % in men at high dosages.
• Flumedroxone acetate is said to have weak or slight progestogenic activity without other hormonal activity ( including estrogenic, antiestrogenic, androgenic, anabolic, or glucocorticoid ).
• At the AR, oxendolone is not a silent antagonist but is rather predominantly antagonistic with weak agonistic activity; The drug has antigonadotropic properties via its progestogenic actions.
• These contraceptives inconsistently inhibit ovulation in ~ 50 % of cycles and rely mainly on their progestogenic effect of thickening the cervical mucus and thereby reducing sperm viability and penetration.